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BET Isoform Selectivity through Diverse Linkers for Bivalent Inhibitors: GSK785, a BRD2/4-Selective Bivalent BET Inhibitor

Lookup NU author(s): Dr Kallie FristonORCiD

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Author(s): Rianjongdee F, Atkinson SJ, Bamborough P, Barnett HA, Friston K, Grandi P, Neipp CE, Petretich M, Phillipou A, Preston AGS, Prinjha RK, Tomkinson NCO, Demont EH

Publication type: Article

Publication status: Published

Journal: Journal of Medicinal Chemistry

Year: 2025

Volume: 69

Issue: 2

Pages: 895-917

Print publication date: 22/01/2026

Online publication date: 30/12/2025

Acceptance date: 19/12/2025

ISSN (print): 0022-2623

ISSN (electronic): 1520-4804

Publisher: American Chemical Society

URL: https://doi.org/10.1021/acs.jmedchem.5c00622

DOI: 10.1021/acs.jmedchem.5c00622

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