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Synthesis of a 3-aminopiperidin-2,5-dione as a conformationally constrained surrogate of the Ala-Gly dipeptide

Lookup NU author(s): Professor Richard Jackson

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Abstract

The preparation of the Boc-{Ala-Gly}-OBn pseudopeptide 4 is reported. The key intermediate, aminoester 5b, was obtained by a cross-coupling reaction of alaninezinc iodide 6 and the thioester of glycine 9. © 2000 Elsevier Science Ltd.

Publication metadata

Author(s): Estiarte MA, Diez A, Rubiralta M, Jackson RFW

Publication type: Article

Publication status: Published

Journal: Tetrahedron

Year: 2001

Volume: 57

Issue: 1

Pages: 157-161

ISSN (print): 0040-4020

ISSN (electronic): 1464-5416

Publisher: Pergamon

URL: http://dx.doi.org/10.1016/S0040-4020(00)00990-X

DOI: 10.1016/S0040-4020(00)00990-X

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